Rankings / Cognitive — Prescription Stimulants

Ephedrine / pseudoephedrine / synephrine stimulants

Cognitive · Sympathomimetic stimulant

Tier C

High-risk evidence profile

wadastimulantsympathomimeticbanned-sport
High-risk evidence profile
4.9 / 10
Tier C
Ev 6 Bn 5 Sf 3.5

Bottom line

Read Off Label grades Ephedrine / pseudoephedrine / synephrine stimulants as C (4.9/10) based on moderate evidence, med benefit magnitude, and a med-high-risk safety profile.

Its high-risk evidence profile reflects a Safety score of 3.5/10; reported benefits and harms can differ by indication, dose, route, duration, and population.

WADA coverage: ephedrine, methylephedrine, pseudoephedrine, cathine, phenylephrine, phenylpropanolamine and synephrine-related stimulant use.

Studied, labeled, or reported-use context: Clinical decongestant/bronchodilator dosing varies; no performance dose — OTC/Rx/status varies; ephedrine and pseudoephedrine are WADA S6 prohibited in competition above thresholds; synephrine is monitoring/not prohibited; not individualized guidance.

What the evidence says

WADA coverage: ephedrine, methylephedrine, pseudoephedrine, cathine, phenylephrine, phenylpropanolamine and synephrine-related stimulant use. Synephrine is included because it appears in WADA monitoring and is common in fat-loss supplement stacks, not because it is prohibited in 2026.

Mechanism

Ephedrine-family sympathomimetics raise adrenergic tone and are used for alertness, nasal decongestion and historically fat loss; thresholds and permitted status differ by compound and dose.

Studied, labeled, or reported dose & route

Clinical decongestant/bronchodilator dosing varies; no performance dose

This records doses and routes described in studies, approved labeling, clinical practice, or documented use. It is not individualized guidance and does not establish safety; context changes with indication, formulation, health history, monitoring, and other medicines.

Citations

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Common questions

What does the evidence show about Ephedrine / pseudoephedrine / synephrine stimulants's effects?
Read Off Label rates the evidence for Ephedrine / pseudoephedrine / synephrine stimulants as Moderate and the benefit magnitude as med, producing an overall grade of C (4.9/10). WADA coverage: ephedrine, methylephedrine, pseudoephedrine, cathine, phenylephrine, phenylpropanolamine and synephrine-related stimulant use.
What safety findings are reported for Ephedrine / pseudoephedrine / synephrine stimulants?
Ephedrine / pseudoephedrine / synephrine stimulants has a med-high risk profile in the database. Med-High (BP/HR elevation, arrhythmia/stroke risk at high dose or combinations, anxiety/insomnia) Legal status: OTC/Rx/status varies; ephedrine and pseudoephedrine are WADA S6 prohibited in competition above thresholds; synephrine is monitoring/not prohibited.
What does the low Safety score for Ephedrine / pseudoephedrine / synephrine stimulants represent?
The Safety score is 3.5/10. It records the substantial harms described for one or more use contexts; the Benefit score, indication, dose, route, duration, population, and legal status remain separate parts of the evidence profile.
What doses or routes are reported for Ephedrine / pseudoephedrine / synephrine stimulants?
Clinical decongestant/bronchodilator dosing varies; no performance dose This is context from studies, approved labeling, clinical practice, or documented use; it is not individualized guidance and does not establish safety.
How does Ephedrine / pseudoephedrine / synephrine stimulants work?
Ephedrine-family sympathomimetics raise adrenergic tone and are used for alertness, nasal decongestion and historically fat loss; thresholds and permitted status differ by compound and dose.

This is an independent synthesis of published research by a non-clinician. Scores are opinions supported by citations, not prescriptions. See the full disclaimer and methodology for how this score was produced and what it does and doesn't mean.