Rankings / Hormones & Endocrine

Gonadorelin (GnRH)

Hormones & Endocrine · Pulsatile GnRH analog

Tier B+

peptidegnrh-axisprescription
7.2 / 10
Tier B+
Ev 8 Bn 5 Sf 7

Bottom line

Read Off Label grades Gonadorelin (GnRH) as B+ (7.2/10) based on strong evidence, med benefit magnitude, and a low-med-risk safety profile.

Becoming the go-to HCG replacement at US men's-health telehealth clinics due to HCG supply disruption and counterfeits.

Studied, labeled, or reported-use context: TRT adjunct: 100-200 mcg subQ 2-3x/week — Rx (LutrePulse discontinued; now compounded); Category 1 on 503A bulks — compounding allowed; not individualized guidance.

What the evidence says

Becoming the go-to HCG replacement at US men's-health telehealth clinics due to HCG supply disruption and counterfeits. Very short half-life (~2-4 min) means subQ injection gives a brief pulse similar to physiological signaling. Listed by FDA as Category 1 (compounding allowed) unlike most other peptides.

Mechanism

Synthetic GnRH identical to endogenous hypothalamic decapeptide; stimulates pituitary LH/FSH when delivered pulsatilely; continuous delivery paradoxically desensitizes pituitary

Studied, labeled, or reported dose & route

TRT adjunct: 100-200 mcg subQ 2-3x/week

This records doses and routes described in studies, approved labeling, clinical practice, or documented use. It is not individualized guidance and does not establish safety; context changes with indication, formulation, health history, monitoring, and other medicines.

Citations

A link means the source informed this entry; it does not mean every claim on the page comes from that source. If a citation looks wrong or you want a claim re-checked, send a correction.

Common questions

What does the evidence show about Gonadorelin (GnRH)'s effects?
Read Off Label rates the evidence for Gonadorelin (GnRH) as Strong and the benefit magnitude as med, producing an overall grade of B+ (7.2/10). Becoming the go-to HCG replacement at US men's-health telehealth clinics due to HCG supply disruption and counterfeits.
What safety findings are reported for Gonadorelin (GnRH)?
Gonadorelin (GnRH) has a low-med risk profile in the database. Low-Med (injection site; ovarian hyperstimulation syndrome in women on fertility doses; desensitization if not dosed correctly) Legal status: Rx (LutrePulse discontinued; now compounded); Category 1 on 503A bulks — compounding allowed.
What doses or routes are reported for Gonadorelin (GnRH)?
TRT adjunct: 100-200 mcg subQ 2-3x/week This is context from studies, approved labeling, clinical practice, or documented use; it is not individualized guidance and does not establish safety.
How does Gonadorelin (GnRH) work?
Synthetic GnRH identical to endogenous hypothalamic decapeptide; stimulates pituitary LH/FSH when delivered pulsatilely; continuous delivery paradoxically desensitizes pituitary

This is an independent synthesis of published research by a non-clinician. Scores are opinions supported by citations, not prescriptions. See the full disclaimer and methodology for how this score was produced and what it does and doesn't mean.