Rankings / Hormones & Endocrine

Pyrilutamide (KX-826)

Hormones & Endocrine · Topical androgen receptor antagonist

Tier C

androgen-receptortopicalagainvestigational
4.9 / 10
Tier C
Ev 3 Bn 5 Sf 7

Bottom line

Read Off Label grades Pyrilutamide (KX-826) as C (4.9/10) based on weak evidence, med benefit magnitude, and a low-med-risk safety profile.

Kintor Pharmaceutical.

Typical use: Topical, applied to scalp twice daily — Investigational.

What this is

Kintor Pharmaceutical. Topical AR antagonist for AGA: China Phase 3 ongoing; US Phase 2 results mixed (inconsistent primary endpoints), Phase 3 design under revision. Mechanistically similar to topical clascoterone. Industry-sponsored; not yet conclusive.

Mechanism

Topical androgen-receptor antagonist for androgenetic alopecia, blocking scalp DHT signaling locally to avoid the systemic sexual side effects of oral finasteride/dutasteride.

Dose & route

Topical, applied to scalp twice daily

Citations

Links go to the source. If a link is dead or you want something re-checked, let me know.

Common questions

Does Pyrilutamide (KX-826) work?
Read Off Label rates the evidence for Pyrilutamide (KX-826) as Weak and the benefit magnitude as med, producing an overall grade of C (4.9/10). Kintor Pharmaceutical.
Is Pyrilutamide (KX-826) safe?
Pyrilutamide (KX-826) has a low-med risk profile in published human data. Legal status: Investigational (China Phase 3; US Phase 2/3). This is not medical advice — see the disclaimer.
What is the typical dose for Pyrilutamide (KX-826)?
Topical, applied to scalp twice daily
How does Pyrilutamide (KX-826) work?
Topical androgen-receptor antagonist for androgenetic alopecia, blocking scalp DHT signaling locally to avoid the systemic sexual side effects of oral finasteride/dutasteride.

This is an independent synthesis of published research by a non-clinician. Scores are opinions supported by citations, not prescriptions. See the full disclaimer and methodology for how this score was produced and what it does and doesn't mean.